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GLL 398
CAS No. 2077980-80-2
GLL 398 ( —— )
产品货号. M29017 CAS No. 2077980-80-2
GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥3540 | 有现货 |
|
| 10MG | ￥5306 | 有现货 |
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| 25MG | ￥9542 | 有现货 |
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| 50MG | ￥14321 | 有现货 |
|
| 100MG | ￥21481 | 有现货 |
|
| 200MG | ￥32222 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称GLL 398
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.
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产品描述GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.(In Vitro):GLL398 exhibits a strong dose-dependent binding profile for the estrogen receptor with a Y537S point mutation with an IC50 of 29.5 nM.
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同义词——
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体Estrogen Receptor/ERR
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研究领域——
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适应症——
化学信息
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CAS Number2077980-80-2
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分子量398.3
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分子式C25H23BO4
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纯度>98% (HPLC)
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溶解度——
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SMILES——
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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